Groups
Year
Paper
2024
Probing the Chemical Space of Guanidino-Carboxylic Acids to Identify the First Blockers of the Creatine-Transporter-1
Clemens V Farr, Yi Xiao, Ali El-Kasaby, Manuel Schupp, Matej Hotka, Giovanni di Mauro, Amy Clarke, Miryam Pastor Fernandez, Walter Sandtner, Thomas Stockner, Christoph Klade, Nuno Maulide, Michael Freissmuth.Mol Pharmacol. 2024 Nov 18;106(6):319-333. doi: 10.1124/molpharm.124.000995.
Abstract: https://pubmed.ncbi.nlm.nih.gov/39322412/
2024
Diastereoselective hydride transfer enables a synthesis of chiral 1,5-carboxamido-trifluoromethylcarbinols
Roberto Tinelli, Manuel Schupp, Immo Klose, Saad Shaaban, Boris Maryasin, Leticia González, Nuno Maulide.Chem Sci. 2024 Sep 9;15(38):15751-6. doi: 10.1039/d4sc05049e. Online ahead of print.
Abstract: https://pubmed.ncbi.nlm.nih.gov/39263662/
2024
Domino Conjugate Addition-1,4-Aryl Migration for the Synthesis of α,β-Difunctionalized Amides
Haoqi Zhang, Yi Xiao, Miran Lemmerer, Tommaso Bortolato, Nuno Maulide.JACS Au. 2024 Jun 17;4(7):2456-2461. doi: 10.1021/jacsau.4c00378. eCollection 2024 Jul 22.
Abstract: https://pubmed.ncbi.nlm.nih.gov/39055149/
2024
PyrAtes: Modular Organic Salts with Large Stokes Shifts for Fluo-rescence Microscopy
Iakovos Saridakis, Margaux Riomet, Oliver J V Belleza, Guilhem Coussanes, Nadja K Singer, Nina Kastner, Yi Xiao, Elliot Smith, Veronica Tona, Aurélien de la Torre, Eric F Lopes, Pedro A Sánchez-Murcia, Leticia González, Harald H Sitte, Nuno Maulide.Angew Chem Int Ed Engl. 2024 May 6;63(19):e202318127. doi: 10.1002/anie.202318127. Epub 2024 Apr 3.
Abstract: https://pubmed.ncbi.nlm.nih.gov/38570814/
2023
Mechanistic Study on Selenium- and Sulfur-Mediated Isomerization of Hydroxamic Acids
Ricardo Meyrelles, Manuel Schupp, Boris Maryasin.Chemistry. 2023 Dec 19;29(71):e202302386. doi: 10.1002/chem.202302386. Epub 2023 Nov 5.
Abstract: https://pubmed.ncbi.nlm.nih.gov/37769009/
2022
Synthesis of α-Aryl Acrylamides via Lewis-Base-Mediated Aryl/Hydrogen Exchange
Miran Lemmerer, Haoqi Zhang, Anthony J Fernandes, Tobias Fischer, Marianne Mießkes, Yi Xiao, Nuno Maulide.Angew Chem Int Ed Engl. 2022 Oct 4;61(40):e202207475. doi: 10.1002/anie.202207475. Epub 2022 Aug 29.
Abstract: https://pubmed.ncbi.nlm.nih.gov/35881564/
Year
Paper
2021
Chuang HY, Schupp M, Meyrelles R, Maryasin B, Maulide N. Redox-Neutral Selenium-Catalysed Isomerisation of para-Hydroxamic Acids into para-Aminophenols. Angew Chem Int Ed Engl. 2021 Mar 24. doi: 10.1002/anie.202100801. Online ahead of print.
Abstract: https://pubmed.ncbi.nlm.nih.gov/33760338/
Abstract: https://pubmed.ncbi.nlm.nih.gov/33760338/
2020
Porte V, Di Mauro G, Schupp M, Kaiser D, Maulide N. Chemoselective Alpha-Deuteration of Amides via Retro-ene Reaction. Chemistry. 2020 Dec 1;26(67):15509-15512. doi: 10.1002/chem.202004103. Epub 2020 Nov 17.
Abstract: https://pubmed.ncbi.nlm.nih.gov/33035360/
Abstract: https://pubmed.ncbi.nlm.nih.gov/33035360/
2019
Chen Y, Coussanes G, Souris C, Aillard P, Kaldre D, Runggatscher K, Kubicek S, Di Mauro G, Maryasin B, Maulide N. A Domino 10-Step Total Synthesis of FR252921 and Its Analogues, Complex Macrocyclic Immunosuppressants. J Am Chem Soc. 2019 Sep 4;141(35):13772-13777. doi: 10.1021/jacs.9b07185.
Abstract: https://pubmed.ncbi.nlm.nih.gov/31436963/
Abstract: https://pubmed.ncbi.nlm.nih.gov/31436963/